Adverse event | Group A2(n=9) | Group B3(n=6) | Group C4(n=21) | Group D5(n=6) | ||||
---|---|---|---|---|---|---|---|---|
Gd 3 | Gd 4 | Gd 3 | Gd 4 | Gd 3 | Gd 4 | Gd 3 | Gd 4 | |
Fatigue | 2 | - | - | - | 6 | - | 2 | 2 |
Febrile neutropenia | - | 3 | 2 | - | 1 | - | - | - |
Alopecia | - | - | - | - | 3 | - | - | - |
Nausea | 1 | - | - | - | 1 | - | - | - |
Respiratory infection | - | - | 1 | - | - | - | 1 | - |
Vomiting | - | - | - | - | 2 | - | - | - |
Anaemia | - | - | - | - | 1 | - | - | - |
Anorexia | - | - | - | - | 1 | - | - | - |
Dehydration | - | - | - | - | 1 | - | - | - |
Diarrhoea | - | - | - | - | 1 | - | - | - |
Leukopenia | 1 | - | - | - | - | - | - | - |
QT/QTc prolongation | - | - | - | - | - | - | 1 | - |
Weight loss | - | - | - | - | 1 | - | - | - |